Friday, 8 May 2020

Reversatol in endometriosis -a new agent



Resveratrol  in Endometriosis and as an alternative agent  to suppress endometriotic lesion :--The solo reason is that, wine contains small amounts of resveratrol, <1-2 mg/8 ounces of red wine and that molecules prevents cancer and ameliorates endometriosis progression.. Red wine has more resveratrol than white wine because red wines are fermented with the grape skins longer than white wines. Hence, many of the antioxidants including resveratrol that are naturally present in the grape skins are extracted into the wine.


How effective is Reversatolol on suppressive  effects on of endometriosis lesion  growth by Reversatolol can be concurrently prescribed with Drospirenone containg OCP. While using a continuous regimen of a combined pill containing drospirenone and ethinyl estradiol, the concomitant use of resveratrol at a daily dose of 30 mg resulted in a significant reduction in the number of patients reporting the occurrence of pain. Growing evidence indicates that this compound possesses A) antineoplastic,B)  anti-inflammatory


and C) antioxidant properties. Resveratrol is a potent D) inhibitor of vascularization in endometriotic lesions
 .E) Resveratrol is a pleiotropic agent, which dose- dependently suppresses the development of new blood vessels. All these properties collectively, cause the suppression of endometriosis lesion growth.

 Effect on cancer Besides having documente effect o endometriosis , Resveratrol has also been shown to exhibit profound in vitro and in vivo G) Effect on cancer :-Growth inhibiting and apoptosis - inducing activities in several biological systems, cancer cell lines and animal models of carcinogenesis. These properties have been linked to inhibition of proliferation in association with cell cycle arrest and, in some systems, with increased apoptotic cell death. Mechanisms of action of resveratrol further include multiple cellular targets affecting various signal transduction pathways, including AKT, RPS6KB2 (p70S6K), mitogen-activated protein kinase 1/3 (MAPK1/3; ERK1/2), STAB, MAPK14 (P38), protein kinase C and peroxisome proliferator-activated receptors (PPARs)-gamma. Importantly, several of these pathways arc relevant to the pathophysiology of endometriosis


Wherefrom we can get Resveratrol:-Resveratrol is also present in the seeds and pomace of grapes . R
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What are new agents for endometriosis?? Anti angiogenic agents of different substance groups are currently discussed as promising candidates for future endometriosis therapy. Besides specific 1)  growth factor antagonists, 2)  endogenous angiogenesis inhibitors, 3) statins, 4) cyclooxygenase-2 inhibitors and 5) other immunomodulators, exert  antiangiogenic effects  ,In this category 6)  also include several phytochemical compounds. The latter ones have been successfully used in traditional medicine without inducing severe side effects what extent there is  association between endometriosis and infertility is still undefined .The medical therapy for endometriosis is symptomatic rather than curative and most patients experience pain relapse at suspension of treatment because restoration of ovulation and of physiological levels of estrogen restore the metabolic activity of both eutopic and ectopic endometrium.

Unfortunately, these approaches often have only modest success and are associated with significant risk of complications and side effects; consequently, the search continues for new, safe and effective long-term treatments. This leads to development of newer modalities in the management of disease.

The often subtle and varied appearances of endometriosis can make recognition and surgical staging difficult, thereby casting doubt on the utility of the classification systems that have been developed. Nevertheless, the findings of well-designed clinical trials and recent studies that elucidated the pathogenesis of endometriosis have enabled a more rational approach to the medical and surgical management of endometriosis.

. Thus, in view of their favorable risk profile, they may be also highly preferable for the safe treatment of endometriosis patients .

However, the association between endometriosis and infertility is still undefined, and there are scanty data to support the many hormonal and surgical therapies that have been proposed. All these controversies and uncertainties have led to use of certain unconventional or less documented therapies, which may be helpful in managing the disease or preventing the complications..
It is widely accepted that peritoneal endometriotic lesions develop from endometrial tissue fragments, which are retrogradly shed through the fallopian tubes during menstruation. During the past few years, numerous studies could demonstrate that the establishment and survival of these lesions is crucially dependent on the formation of blood vessels, which guarantee their oxygen supply. Accordingly, -
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Resveratrol is one such natural phytoalexin, which represents one of the most frequently analysed phytochemical compounds in life sciences during the last decades. phytochemical treatment of endometriosis. Because resveratrol exerts a broad spectrum of beneficial effects under various pathological conditions, it has been suggested as a promising therapeutic agent for the treatment of cancer as well as several inflammatory, metabolic and cardiovascular diseases.
Resveratrol is a polyphenol synthesized by plants following ultraviolet radiation and fungal infections. Resveratrol (3,5,4’-trihydroxy-trans-stilbene) is found in red grape skin, Japanese knotweed (Polygonum cuspidatum), peanuts, blueberries and some other berries. A large amount of resveratrol is produced in the skin of grapes to protect the plant against fungal diseases and sun damage; therefore, wine has higher levels of resveratrol compared to other natural food. Overall, red wine contains small amounts of resveratrol, <1-2 mg/8 ounces of red wine. However, red wine has more resveratrol than white wine because red wines are fermented with the grape skins longer than white wines. Hence, many of the antioxidants including resveratrol that are naturally present in the grape skins are extracted into the wine. Resveratrol is also present in the seeds and pomace of grapes

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